Celastrol CAS 34157-83-0
Celastrol ntishobora gushonga mumazi, gushonga muri dimethyl sulfoxide na Ethanol ya anhydrous. Bikomoka ku kurwanya kanseri ikora mu bimera nka Thunder God Vine na Vine Inzoka y'Amajyepfo mu muryango Celastraceae. Inzitizi nziza ya proteasome, yemejwe gutera kanseri ya apoptose ya kanseri ihagarika ibikorwa bya proteasome
Ingingo | Ibisobanuro |
Ingingo yo guteka | 645.7 ± 55.0 ° C (Biteganijwe) |
Ubucucike | 1.2 |
Ingingo yo gushonga | 219-230 ° C. |
pKa | 4.78 ± 0.70 (Byahanuwe) |
xmax | 424nm (MeOH) (lit.) |
Imiterere yo kubika | -20 ° C. |
Celastrol ikoreshwa muguhitamo ibirimo / kumenyekanisha / ubushakashatsi bwa farumasi, nibindi. Ingaruka za farumasi: Ifite antioxydants ikomeye, anti-kanseri angiogenezi, na anti-rheumatoide. Inzitizi nziza ya proteasome, yemejwe gutera kanseri ya apoptose ya kanseri ihagarika ibikorwa bya proteasome
Mubisanzwe bipakiye muri 25kg / ingoma, kandi birashobora no gukora pake yabigenewe.

Celastrol CAS 34157-83-0

Celastrol CAS 34157-83-0